Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain

Michael Brand, James Clayton, Mustafa Moroglu, Matthias Schiedel, Sarah Picaud, Joseph P. Bluck, Anna Skwarska, Hannah Bolland, Anthony K.N. Chan, Corentine M.C. Laurin, Amy R. Scorah, Larissa See, Timothy P.C. Rooney, Katrina H. Andrews, Oleg Fedorov, Gabriella Perell, Prakriti Kalra, Kayla B. Vinh, Wilian A. Cortopassi, Pascal HeitelKirsten E. Christensen, Richard I. Cooper, Robert S. Paton, William C.K. Pomerantz, Philip C. Biggin, Ester M. Hammond, Panagis Filippakopoulos, Stuart J. Conway

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